SCHEMBL7894178

SCHEMBL7894178

COc1cc(C#N)ccc1CNc1c(NC(C)C(C)(C)C)c(=O)c1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 1/20 0.58
ABCC8 Q09428 1/20 0.58
KCNJ11 Q14654 1/20 0.58
KCNJ8 Q15842 1/20 0.58
PLK1 P53350 8/20 0.43
GSK3A P49840 3/20 0.43
ROCK1 Q13464 3/20 0.43
CDC42BPA Q5VT25 3/20 0.43
RPS6KB1 P23443 2/20 0.43
AURKB Q96GD4 2/20 0.43
GSK3B P49841 2/20 0.43
CSNK1G3 Q9Y6M4 2/20 0.43
ERBB2 P04626 1/20 0.43
PRKACA P17612 1/20 0.43
IRAK1 P51617 1/20 0.43
RPS6KA3 P51812 1/20 0.43
CHEK1 O14757 3/20 0.42
MAPK1 P28482 3/20 0.42
PLK4 O00444 2/20 0.42
DAPK3 O43293 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7887074 0.85 ABCC9 (0.71) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL7895748 0.85 ABCC9 (0.61) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL7895113 0.84 ABCC9 (0.60) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL7895591 0.84 ABCC9 (0.60) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL8670505 0.82 ABCC9 (0.70) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL8670509 0.82 ABCC9 (0.70) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL7886866 0.78 ABCC9 (0.58) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL7886860 0.78 ABCC9 (0.58) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL7894022 0.78 ABCC9 (0.58) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL7894099 0.76 ABCC9 (0.50) ABCC9ABCC8KCNJ11KCNJ8GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1151990-A1 Substituted N-arylmethylamino derivatives of cyclobutene-3, 4-diones AMERICAN HOME PRODUCTS CORPORATION (US) 2001-11-07 EP claimed
US-5780505-A ADMINISTERING AS SMOOTH MUSCLE RELAXANT AMERICAN HOME PRODUCTS CORPORATION (US) 1998-07-14 US claimed
EP-1151990-A1 Substituted N-arylmethylamino derivatives of cyclobutene-3, 4-diones AMERICAN HOME PRODUCTS CORPORATION (US) 2001-11-07 EP disclosed
US-5780505-A ADMINISTERING AS SMOOTH MUSCLE RELAXANT AMERICAN HOME PRODUCTS CORPORATION (US) 1998-07-14 US disclosed