SCHEMBL789462

SCHEMBL789462

COc1ccc(S(=O)(=O)Nc2cc(B3OC(C)(C)C(C)(C)O3)cnc2OC)cc1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPL P05186 1/20 0.49
KEAP1 Q14145 1/20 0.47
NFE2L2 Q16236 1/20 0.47
ALDH1A1 P00352 3/20 0.46
TP53 P04637 1/20 0.46
ABCB1 P08183 1/20 0.46
ABCC1 P33527 1/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
MAPK1 P28482 1/20 0.46
LMNA P02545 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
HTT P42858 1/20 0.45
PKM P14618 1/20 0.44
CA12 O43570 1/20 0.44
CA9 Q16790 1/20 0.44
EDNRA P25101 2/20 0.43
FFAR4 Q5NUL3 1/20 0.43
CYP2C9 P11712 1/20 0.42
EDNRB P24530 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15462778 0.87 ALPL (0.51) ALPLKEAP1NFE2L2ALDH1A1MEN1
SCHEMBL15459550 0.87 ALPL (0.51) ALPLTP53MEN1KMT2ALMNA
SCHEMBL22447720 0.87 ALPL (0.48) ALPLALDH1A1ABCB1ABCC1MEN1
SCHEMBL15559069 0.86 ALPL (0.52) ALPLALDH1A1
SCHEMBL15650005 0.86 ALPL (0.50) ALPLCA9
SCHEMBL22508714 0.86 ALPL (0.50) ALPLALDH1A1TP53LMNAHTT
SCHEMBL790824 0.86 ALPL (0.56) ALPL
SCHEMBL29556839 0.86 ALPL (0.56) ALPL
SCHEMBL28554047 0.85 ALPL (0.51) ALPL
SCHEMBL15649752 0.85 ALPL (0.47) ALPLALDH1A1MEN1KMT2ACA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012174312-A2 BENZIMIDAZOLE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-12-20 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed