SCHEMBL7895461

SCHEMBL7895461

CCOC(=O)C1C2CN(C(=O)OC(C)(C)C)CC21

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.48
MEN1 O00255 2/20 0.42
ALDH1A1 P00352 2/20 0.42
KMT2A Q03164 2/20 0.42
TSHR P16473 1/20 0.42
SSTR4 P31391 1/20 0.41
MAPT P10636 2/20 0.39
USP2 O75604 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GPR119 Q8TDV5 2/20 0.38
NAMPT P43490 1/20 0.38
JAK3 P52333 1/20 0.38
ADORA1 P30542 1/20 0.38
HPGD P15428 1/20 0.37
PPM1B O75688 1/20 0.36
PTPN1 P18031 1/20 0.36
PPP1CC P36873 1/20 0.36
PDE4B Q07343 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16252085 1.00 NR1H2 (0.48) NR1H2MEN1ALDH1A1KMT2ATSHR
SCHEMBL31554278 1.00 NR1H2 (0.48) NR1H2MEN1ALDH1A1KMT2ATSHR
SCHEMBL12277546 1.00 NR1H2 (0.48) NR1H2MEN1ALDH1A1KMT2ATSHR
SCHEMBL29928249 1.00 NR1H2 (0.48) NR1H2MEN1ALDH1A1KMT2ATSHR
SCHEMBL17387946 1.00 NR1H2 (0.48) NR1H2MEN1ALDH1A1KMT2ATSHR
SCHEMBL15890054 1.00 NR1H2 (0.48) NR1H2MEN1ALDH1A1KMT2ATSHR
SCHEMBL25394396 0.90 ALDH1A1 (0.46) NR1H2MEN1ALDH1A1KMT2ATSHR
SCHEMBL12615290 0.84 ALDH1A1 (0.50) NR1H2MEN1ALDH1A1KMT2ATSHR
SCHEMBL1052491 0.84 NR1H2 (0.50) NR1H2MEN1ALDH1A1KMT2ATSHR
SCHEMBL2930651 0.84 NR1H2 (0.50) NR1H2MEN1ALDH1A1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12448368-B2 Indole compounds as androgen receptor modulators NIDO BIOSCIENCES, INC. (US) 2025-10-21 US disclosed
US-20250122176-A1 INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS NIDO BIOSCIENCES INC (US) 2025-04-17 US disclosed
US-20250092021-A9 INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS NIDO BIOSCIENCES, INC. 2025-03-20 US disclosed
WO-2025039774-A1 IMIDAZO[1,2-A]PYRIDINE TYPE IRAK DEGRADATION AGENT AND USE THEREOF 泰诺瑞(天津)生物科技有限责任公司 2025-02-27 WO disclosed
CN-118955497-A Imidazo [1,2-a ] pyridine IRAK4 degradation agent and application thereof 泰诺瑞(天津)生物科技有限责任公司 2024-11-15 CN disclosed
US-20230348439-A1 INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS NIDO BIOSCIENCES INC (US) 2023-11-02 US disclosed
US-11667624-B2 Indole compounds as androgen receptor modulators NIDO BIOSCIENCES, INC. (US) 2023-06-06 US disclosed
EP-4182320-A1 INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS Nido Biosciences, Inc. (US) 2023-05-24 EP disclosed
US-20230049406-A1 INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS NIDO BIOSCIENCES, INC. 2023-02-16 US disclosed
WO-2022109551-A1 SRC INHIBITORS AND USES THEREOF RELAY THERAPEUTICS, INC. (US) 2022-05-27 WO disclosed
US-8895602-B1 6-pyrazolylamido-3-substituted azabicyclo[3.1.0]hexane compounds as calcium channel inhibitors KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2014-11-25 US disclosed
US-8895602-B1 6-pyrazolylamido-3-substituted azabicyclo[3.1.0]hexane compounds as calcium channel inhibitors KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2014-11-25 US disclosed
US-20140343295-A1 NOVEL 6-PYRAZOLYLAMIDO-3-SUBSTITUTED AZABICYCLO[3.1.0]HEXANE COMPOUNDS AS CALCIUM CHANNEL INHIBITORS KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2014-11-20 US disclosed
US-20140343295-A1 NOVEL 6-PYRAZOLYLAMIDO-3-SUBSTITUTED AZABICYCLO[3.1.0]HEXANE COMPOUNDS AS CALCIUM CHANNEL INHIBITORS KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2014-11-20 US disclosed
US-8497289-B2 3.1.0 bicyclic GlyT1 inhibitors and methods of making and using same VANDERBILT UNIVERSITY (US) 2013-07-30 US disclosed
US-8497289-B2 3.1.0 bicyclic GlyT1 inhibitors and methods of making and using same VANDERBILT UNIVERSITY (US) 2013-07-30 US disclosed
US-8497289-B2 3.1.0 bicyclic GlyT1 inhibitors and methods of making and using same VANDERBILT UNIVERSITY (US) 2013-07-30 US disclosed
US-20100256192-A1 3.1.0 BICYCLIC GLYT1 INHIBITORS AND METHODS OF MAKING AND USING SAME VANDERBILT UNIVERSITY 2010-10-07 US disclosed
US-20100256192-A1 3.1.0 BICYCLIC GLYT1 INHIBITORS AND METHODS OF MAKING AND USING SAME VANDERBILT UNIVERSITY 2010-10-07 US disclosed
WO-2010078348-A1 3.1.0 BICYCLIC GLYT1 INHIBITORS AND METHODS OF MAKING AND USING SAME VANDERBILT UNIVERSITY (US) 2010-07-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230049406-A1 INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS AR, FSHR, NR5A1 NR1H2 86/4885MEN1 2818/4885ALDH1A1 2325/4885
US-20230348439-A1 INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS AR, FSHR, NR5A1 NR1H2 88/4885MEN1 2673/4885ALDH1A1 2260/4885
US-20250122176-A1 INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS AR, FSHR, NR5A1 NR1H2 86/4885MEN1 2818/4885ALDH1A1 2325/4885
US-11667624-B2 Indole compounds as androgen receptor modulators AR, FSHR, ADRB3 NR1H2 134/4885MEN1 2646/4885ALDH1A1 2697/4885
US-20250092021-A9 INDOLE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS AR, FSHR, NR5A1 NR1H2 86/4885MEN1 2818/4885ALDH1A1 2325/4885
US-20140343295-A1 NOVEL 6-PYRAZOLYLAMIDO-3-SUBSTITUTED AZABICYCLO[3.1.0]HEXANE COMPOUNDS AS CALCIUM CHANNEL INHIBITORS CACNA1B, CACNA1I, CACNA1D NR1H2 3353/4885MEN1 1174/4885ALDH1A1 3014/4885
US-12448368-B2 Indole compounds as androgen receptor modulators AR, FSHR, ADRB3 NR1H2 134/4885MEN1 2646/4885ALDH1A1 2697/4885
US-20100256192-A1 3.1.0 BICYCLIC GLYT1 INHIBITORS AND METHODS OF MAKING AND USING SAME SLC7A1, SLC5A1, SLC1A1 NR1H2 1255/4885MEN1 1213/4885ALDH1A1 1138/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.