SCHEMBL789604

SCHEMBL789604

COc1nc(C)c(-c2ccc3nc(N)c(-c4ccc(C(=O)N5CCOCC5)cc4)cc3c2)cc1-c1c(F)ccc(S(N)(=O)=O)c1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 2/20 0.46
PIK3CG P48736 2/20 0.46
KCNH2 Q12809 2/20 0.38
CA2 P00918 2/20 0.36
CA9 Q16790 2/20 0.36
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36
BRD4 O60885 1/20 0.36
GRM2 Q14416 1/20 0.36
JAK2 O60674 2/20 0.35
JAK1 P23458 2/20 0.35
TYK2 P29597 2/20 0.35
JAK3 P52333 2/20 0.35
ERN1 O75460 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MTOR P42345 2/20 0.35
ATR Q13535 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL789483 0.88 PI4KA (0.51) PI4KAPIK3CGKCNH2CA2CA9
SCHEMBL789603 0.81 PIK3CG (0.66) PI4KAPIK3CGMTOR
SCHEMBL789602 0.78 PI4KA (0.41) PI4KAPIK3CGKCNH2CA2CA9
SCHEMBL789482 0.75 PIK3CG (0.65) PI4KAPIK3CGKCNH2MTOR
SCHEMBL791064 0.75 PIK3CG (0.81) PI4KAPIK3CGMTOR
SCHEMBL10277103 0.74 PIK3CG (0.57) PI4KAPIK3CGKCNH2BRD4MTOR
SCHEMBL789481 0.72 PI4KA (0.45) PI4KAPIK3CGKCNH2CA2CA9
SCHEMBL10277220 0.70 PIK3CG (0.78) PI4KAPIK3CGMTOR
SCHEMBL806968 0.70 PIK3CG (0.72) PI4KAPIK3CGMTOR
SCHEMBL791171 0.69 PIK3CG (0.54) PI4KAPIK3CGKCNH2MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed