SCHEMBL7898657

SCHEMBL7898657

CCCC(Br)Oc1ccc(N=C=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.42
TSHR P16473 1/20 0.42
TRPA1 O75762 1/20 0.34
CYP1A2 P05177 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
MAPK1 P28482 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
PPARG P37231 2/20 0.31
PPARA Q07869 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552039 0.75 CA12 (0.44) MAPK1
SCHEMBL6371340 0.75 CYP3A4 (0.46) CYP3A4TSHRTRPA1CYP1A2GABRA1
Butane SCHEMBL16872374 0.74 CYP3A4 (0.62) CYP3A4TSHRTRPA1CYP1A2GABRA1
SCHEMBL11241942 0.74 PPARA (0.41) PPARGPPARA
SCHEMBL9310814 0.74 SLC6A4 (0.41) TSHRCYP1A2TDP1PPARGPPARA
SCHEMBL2773412 0.73 SLC6A4 (0.41) PPARGPPARA
SCHEMBL9111062 0.73 ALDH1A3 (0.53) CYP3A4TSHRTRPA1MAPK1TDP1
SCHEMBL991987 0.73 CYP2C9 (0.50) CYP3A4TSHRCYP1A2MAPK1
SCHEMBL414168 0.73 CYP1A2 (0.50) CYP3A4TSHRCYP1A2
SCHEMBL230798 0.72 NQO1 (0.56) CYP3A4TSHRCYP1A2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999064041-A9 MULTIBINDING AGENTS THAT MODULATE NMDA RECEPTORS ADVANCED MEDICINE INC (US) 2001-05-31 WO disclosed
EP-1100519-A1 MULTIBINDING AGENTS THAT MODULATE NMDA RECEPTORS Advanced Medicine, Inc. (US) 2001-05-23 EP disclosed
WO-1999064041-A1 MULTIBINDING AGENTS THAT MODULATE NMDA RECEPTORS ADVANCED MEDICINE, INC. (US) 1999-12-16 WO disclosed