SCHEMBL7899372

SCHEMBL7899372

CN1C(=O)C2CCC1(C(N[S@+]([O-])C(C)(C)C)c1cccnc1)CC2

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 4/20 0.37
TSHR P16473 2/20 0.35
MAPT P10636 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ITGB3 P05106 2/20 0.33
ITGA2B P08514 2/20 0.33
KDM4E B2RXH2 2/20 0.31
CYP3A4 P08684 1/20 0.31
THRB P10828 1/20 0.31
THPO P40225 1/20 0.31
MEN1 O00255 1/20 0.31
MAPK1 P28482 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CREBBP Q92793 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3707269 1.00 SLC6A9 (0.37) SLC6A9TSHRMAPTHSD17B10ITGB3
SCHEMBL7896578 0.89 SLC6A9 (0.36) SLC6A9
SCHEMBL3708353 0.89 SLC6A9 (0.36) SLC6A9
SCHEMBL4177209 0.88 SLC6A9 (0.36) SLC6A9
SCHEMBL3707332 0.88 SLC6A9 (0.36) SLC6A9
SCHEMBL4177205 0.88 SLC6A9 (0.36) SLC6A9
SCHEMBL3789660 0.78 HTR2A (0.32) ALDH1A1
SCHEMBL3789656 0.78 HTR2A (0.32) ALDH1A1
SCHEMBL3707190 0.77 TSHR (0.41) SLC6A9TSHRMAPTHSD17B10KDM4E
SCHEMBL7899351 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010087761-A1 2-AZA-BICYCLO[2.2.2]OCTANE COMPOUNDS AND USES THEREOF ASTRAZENECA AB (SE) 2010-08-05 WO disclosed