SCHEMBL7899679

SCHEMBL7899679

O=C(N1CCN(c2ccc(F)cc2)CC1)N1CCC(C(=O)NNc2ccc(F)cc2)(c2ccc(F)cc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.51
CA12 O43570 3/20 0.49
CA1 P00915 3/20 0.49
CA2 P00918 3/20 0.49
CA9 Q16790 3/20 0.49
MAPT P10636 6/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
ALOX15 P16050 1/20 0.46
ALOX12 P18054 1/20 0.46
GFER P55789 1/20 0.46
USP2 O75604 1/20 0.45
MAPK1 P28482 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
GLA P06280 1/20 0.44
POLB P06746 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7910246 0.83 AKR1C3 (0.52) AKR1C3CA12CA1CA2CA9
SCHEMBL378652 0.82 AKR1C3 (0.59) AKR1C3CA12CA1CA2CA9
SCHEMBL7908737 0.79 PANK3 (0.48) AKR1C3CA12CA1CA2CA9
SCHEMBL7899677 0.78 AKR1C3 (0.47) AKR1C3CA12CA1CA2CA9
SCHEMBL3107003 0.78 PTPN1 (0.50) RAB9AMEN1KMT2A
SCHEMBL7912655 0.78 PANK3 (0.47) AKR1C3CA12CA1CA2CA9
SCHEMBL13092408 0.78 AKR1C3 (0.46) AKR1C3CA12CA1CA2CA9
SCHEMBL3097422 0.77 NPSR1 (0.61) AKR1C3CA12CA1CA2CA9
SCHEMBL378400 0.76 OPRM1 (0.67) AKR1C3SMN1; SMN2ALDH1A1NPSR1MEN1
SCHEMBL27607283 0.75 AKR1C3 (0.83) AKR1C3CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010106081-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-23 WO disclosed