SCHEMBL7899790

SCHEMBL7899790

Bc1cnc2c(c1)c(-c1ccc3[nH]ccc3c1)cn2S(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.47
TGFBR1 P36897 1/20 0.40
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAP3K11 Q16584 6/20 0.37
LRRK2 Q5S007 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 1/20 0.36
DRD2 P14416 1/20 0.35
HTR6 P50406 1/20 0.35
BRAF P15056 1/20 0.35
PIP4K2A P48426 1/20 0.35
PIP4K2B P78356 1/20 0.35
DYRK1A Q13627 1/20 0.34
DYRK2 Q92630 1/20 0.34
DYRK1B Q9Y463 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL721859 0.89 PTPN11 (0.47) PTPN11TGFBR1CA12CA1CA2
SCHEMBL15171450 0.87 PTPN11 (0.46) PTPN11TGFBR1CA12CA1CA2
SCHEMBL15165532 0.87 PTPN11 (0.46) PTPN11TGFBR1CA12CA1CA2
SCHEMBL7907745 0.85 PTPN11 (0.50) PTPN11TGFBR1MAP3K11LRRK2CYP3A4
SCHEMBL30280395 0.85 PTPN11 (0.51) PTPN11TGFBR1CA12CA1CA2
SCHEMBL721797 0.85 PTPN11 (0.51) PTPN11TGFBR1CA12CA1CA2
SCHEMBL720829 0.83 TGFBR1 (0.41) PTPN11TGFBR1CA12CA1CA2
SCHEMBL15165536 0.83 PTPN11 (0.51) PTPN11TGFBR1CA12CA1CA2
SCHEMBL7899740 0.83 MAP3K11 (0.56) PTPN11MAP3K11LRRK2
SCHEMBL11968502 0.83 PTPN11 (0.44) PTPN11TGFBR1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149950-A2 BICYCLIC HETEROARYL KINASE INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2011-12-01 WO disclosed
WO-2010068483-A2 MLK INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2010-06-17 WO disclosed