SCHEMBL7901172

SCHEMBL7901172

CCCOc1ccccc1-c1nc2c(CCCCc3ccccc3)cccc2c(=O)[nH]1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 19/20 0.56
KDM4E B2RXH2 1/20 0.55
MEN1 O00255 1/20 0.55
PDE2A O00408 1/20 0.55
PDE6D O43924 1/20 0.55
USP2 O75604 1/20 0.55
PDE9A O76083 1/20 0.55
ALDH1A1 P00352 1/20 0.55
LMNA P02545 1/20 0.55
CYP1A2 P05177 1/20 0.55
MAPT P10636 1/20 0.55
HPGD P15428 1/20 0.55
ALOX15 P16050 1/20 0.55
PDE6A P16499 1/20 0.55
PDE6G P18545 1/20 0.55
PDE4A P27815 1/20 0.55
PDE6B P35913 1/20 0.55
PDE6C P51160 1/20 0.55
PDE1A P54750 1/20 0.55
PDE1B Q01064 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7901174 0.98 PDE5A (0.56) PDE5AKDM4EMEN1PDE2APDE6D
SCHEMBL7899533 0.92 PDE5A (0.57) PDE5AKDM4EMEN1PDE2APDE6D
SCHEMBL7901311 0.84 PDE5A (0.52) PDE5AKDM4EMEN1PDE2APDE6D
SCHEMBL7899531 0.83 PDE5A (0.52) PDE5AKDM4EMEN1PDE2APDE6D
SCHEMBL7901179 0.81 PDE5A (0.52) PDE5AKDM4EMEN1PDE2APDE6D
SCHEMBL7159216 0.81 PDE5A (0.66) PDE5AKDM4EMEN1PDE2APDE6D
SCHEMBL7899640 0.81 PDE5A (0.50) PDE5AKDM4EMEN1PDE2APDE6D
SCHEMBL7901175 0.80 PDE5A (0.61) PDE5AKDM4EMEN1PDE2APDE6D
SCHEMBL7901239 0.80 PDE5A (0.61) PDE5AKDM4EMEN1PDE2APDE6D
SCHEMBL7901192 0.80 PDE5A (0.51) PDE5AKDM4EMEN1PDE2APDE6D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187779-B1 ADMINISTERING ANTITUMOR AGENTS TO TREAT COLON CANCER CELL PATHWAYS, INC. 2001-02-13 US disclosed
US-5721238-A ANTIINFLAMMATORY AGENTS, CARDIOVASCULAR DISORDERS BAYER AKTIENGESELLSCHAFT (DE) 1998-02-24 US disclosed
EP-0722937-A1 2,8-Disubstituted quinazolinone BAYER AG (DE) 1996-07-24 EP disclosed