SCHEMBL7901453

SCHEMBL7901453

Cc1ccc(-n2nc3c4ccccc4n(Cc4ccc(-c5ccc(C)nc5)cc4)nc-3c2=O)c(C)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 10/20 0.42
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
F2RL3 Q96RI0 1/20 0.39
FSCN1 Q16658 1/20 0.38
POLB P06746 1/20 0.38
PDE5A O76074 1/20 0.37
TSHR P16473 1/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
PKM P14618 1/20 0.35
PKLR P30613 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3708584 0.91 F2RL3 (0.41) CHRM1ALDH1A1KDM4EF2RL3FSCN1
SCHEMBL3713264 0.79 GABRA1 (0.37) CHRM1F2RL3FSCN1POLBPDE5A
SCHEMBL7913305 0.79 GABRA1 (0.41) CHRM1F2RL3FSCN1POLBPDE5A
SCHEMBL3779687 0.76 GRM2 (0.39) CHRM1ALDH1A1F2RL3FSCN1POLB
SCHEMBL14875518 0.72 GRM2 (0.39) CHRM1ALDH1A1F2RL3FSCN1POLB
SCHEMBL7906411 0.70 FGFR1 (0.47) CHRM1F2RL3
SCHEMBL4478716 0.70 F2RL3 (0.60) ALDH1A1KDM4EF2RL3PDE5AMAPT
SCHEMBL7907818 0.69 PDE5A (0.34) CHRM1ALDH1A1KDM4EF2RL3FSCN1
SCHEMBL3805510 0.69 GRN (0.43) CHRM1FSCN1PDE5AKMT2A
SCHEMBL7909375 0.68 CYP11B1 (0.41) CHRM1ALDH1A1KDM4EPDE5AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010096338-A1 PYRAZOLO [4,3-c] CINNOLIN-3-ONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK SHARP & DOHME CORP. (US) 2010-08-26 WO disclosed