SCHEMBL7902178

SCHEMBL7902178

Cc1ncc(-c2ccc(Cl)s2)o1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.56
CA1 P00915 4/20 0.56
CA2 P00918 4/20 0.56
CA9 Q16790 4/20 0.56
PTGS1 P23219 3/20 0.40
PTGS2 P35354 3/20 0.40
CYP2A6 P11509 1/20 0.40
S1PR4 O95977 1/20 0.39
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
KDM4E B2RXH2 3/20 0.37
HPGD P15428 2/20 0.37
ALDH1A1 P00352 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PDGFRB P09619 1/20 0.36
PDGFRA P16234 1/20 0.36
PIK3CG P48736 1/20 0.36
KDM1A O60341 1/20 0.36
F10 P00742 2/20 0.35
LRRK2 Q5S007 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10053489 0.83 CA12 (0.61) CA12CA1CA2CA9PTGS1
SCHEMBL12545666 0.78 CYP2A6 (0.37) CA12CA1CA2CA9PTGS1
SCHEMBL10022410 0.76 CA12 (0.54) CA12CA1CA2CA9GRIN1
SCHEMBL7503295 0.75 NOTUM (0.37) CA12CA1CA2CA9CYP2A6
SCHEMBL6261333 0.73 CA12 (0.55) CA12CA1CA2CA9KDM4E
SCHEMBL27591541 0.72 NOTUM (0.36) CA12CA1CA2CA9CYP2A6
SCHEMBL27690445 0.69 KDM4E (0.45) CYP2A6KDM4EHPGDALDH1A1F10
SCHEMBL13484009 0.69 ALDH1A1 (0.46) CA12CA1CA2CA9CYP2A6
SCHEMBL7897326 0.69 MAPT (0.48) F10
SCHEMBL7496613 0.69 KDM4E (0.55) CA12CA1CA2CA9PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2373634-B1 MORPHOLINONE COMPOUNDS AS FACTOR IXA INHIBITORS MOCHIDA PHARM CO LTD (JP) 2015-11-11 EP disclosed
WO-2010065717-A1 MORPHOLINONE COMPOUNDS AS FACTOR IXA INHIBITORS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2010-06-10 WO disclosed