SCHEMBL7904072

SCHEMBL7904072

Cc1c(N)cc(Cc2ccccc2)c(C)c1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 1/20 0.45
BCL2L1 Q07817 1/20 0.45
HTR2A P28223 1/20 0.42
CALM1 P0DP23 1/20 0.42
LDHA P00338 1/20 0.42
LDHB P07195 1/20 0.42
ALOX5 P09917 1/20 0.40
CNR2 P34972 1/20 0.39
GPR55 Q9Y2T6 1/20 0.39
LTB4R Q15722 1/20 0.39
USP2 O75604 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
RECQL P46063 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MPO P05164 1/20 0.38
TPO P07202 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28493010 0.89 BCL2 (0.42) BCL2BCL2L1HTR2ACALM1LDHA
SCHEMBL31402366 0.89 BCL2 (0.42) BCL2BCL2L1HTR2ACALM1LDHA
SCHEMBL4649847 0.85 BCL2 (0.40) BCL2BCL2L1HTR2ACALM1LDHA
SCHEMBL10886157 0.85 BCL2 (0.42) BCL2BCL2L1HTR2ACALM1LDHA
SCHEMBL22188467 0.85 BCL2 (0.42) BCL2BCL2L1HTR2ACALM1LDHA
SCHEMBL4650255 0.84 HTR2A (0.42) BCL2BCL2L1HTR2ACALM1ALOX5
SCHEMBL9494600 0.82 BCL2 (0.44) BCL2BCL2L1HTR2ACALM1LDHA
Iodide SCHEMBL22188505 0.82 HTR2A (0.41) BCL2BCL2L1HTR2ACALM1ALOX5
Hydrochloric Acid SCHEMBL1559085 0.82 HTR2A (0.41) BCL2BCL2L1HTR2ACALM1ALOX5
SCHEMBL22232131 0.82 BCL2 (0.44) BCL2BCL2L1HTR2ACALM1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6204337-B1 Solid-phase synthesis of codeine from morphine THE BOARD OF REGENTS OF THE UNIVERSITY AND COMMUNITY COLLEGE SYSTEM OF NEVEDA 2001-03-20 US disclosed
US-5981750-A Solid-phase synthesis of codeine from morphine THE BOARD OF REGENTS OF THE UNIVERSITY AND COMMUNITY COLLEGE SYSTEM OF NEVADA (US) 1999-11-09 US disclosed
WO-1997019082-A1 SOLID-PHASE SYNTHESIS OF CODEINE FROM MORPHINE THE BOARD OF REGENTS OF THE UNIVERSITY AND COMMUNITY COLLEGE SYSTEM OF NEVADA ON BEHALF OF THE UNIVERSITY OF NEVADA-RENO (US) 1997-05-29 WO disclosed