SCHEMBL4649847

SCHEMBL4649847

Cc1c(Cc2ccccc2)cc(N)c(Br)c1C

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 1/20 0.40
BCL2L1 Q07817 1/20 0.40
HTR2A P28223 1/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP1A2 P05177 1/20 0.37
ALOX15 P16050 1/20 0.37
CASP7 P55210 1/20 0.37
HIF1A Q16665 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CALM1 P0DP23 1/20 0.37
CTRC Q99895 1/20 0.37
ALOX5 P09917 1/20 0.36
CNR2 P34972 1/20 0.35
GPR55 Q9Y2T6 1/20 0.35
LDHA P00338 1/20 0.35
LDHB P07195 1/20 0.35
MPO P05164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7904072 0.85 BCL2 (0.45) BCL2BCL2L1HTR2AALDH1A1ALOX15
SCHEMBL31402366 0.82 BCL2 (0.42) BCL2BCL2L1HTR2AALDH1A1ALOX15
SCHEMBL28493010 0.82 BCL2 (0.42) BCL2BCL2L1HTR2AALDH1A1ALOX15
SCHEMBL10886157 0.79 BCL2 (0.42) BCL2BCL2L1HTR2AALDH1A1ALOX15
SCHEMBL9494600 0.77 BCL2 (0.44) BCL2BCL2L1HTR2AALDH1A1ALOX15
SCHEMBL29454271 0.77 BCL2 (0.44) BCL2BCL2L1HTR2ACALM1ALOX5
SCHEMBL22232131 0.77 BCL2 (0.44) BCL2BCL2L1HTR2ACALM1ALOX5
SCHEMBL20159665 0.77 ALDH1A1 (0.55) BCL2BCL2L1HTR2AALDH1A1CYP1A2
SCHEMBL22188467 0.75 BCL2 (0.42) BCL2BCL2L1HTR2AALDH1A1ALOX15
SCHEMBL4650255 0.74 HTR2A (0.42) BCL2BCL2L1HTR2ACALM1CTRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966138-A2 SUBSTITUTED TRICYCLIC PIPERIDONE DERIVATIVES Grünenthal GmbH (DE) 2008-09-10 EP disclosed
WO-2007079929-A2 SUBSTITUTED TRICYCLIC PIPERIDONE DERIVATIVES Grünenthal GmbH (DE) 2007-07-19 WO disclosed