SCHEMBL7904620

SCHEMBL7904620

CC1=C(C#N)[C@@H](c2ccc(C#N)cc2S(C)(=O)=O)n2nc(N)nc2N1c1cccc(C(F)(F)F)c1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ELANE P08246 20/20 0.67
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL230975 1.00 ELANE (0.67) ELANECYP3A4CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL231082 0.99 ELANE (0.66) ELANECYP3A4CYP2C9CYP2C19
SCHEMBL2742318 0.89 ELANE (0.65) ELANECYP2C19
SCHEMBL2742319 0.89 ELANE (0.65) ELANECYP2C19
SCHEMBL15354362 0.87 ELANE (0.50) ELANECYP2C19
SCHEMBL15354374 0.87 ELANE (0.50) ELANECYP2C19
SCHEMBL14632124 0.87 ELANE (0.63) ELANECYP2C19
SCHEMBL230879 0.86 ELANE (0.64) ELANECYP3A4CYP2C9CYP2C19
SCHEMBL230772 0.86 ELANE (0.64) ELANECYP3A4CYP2C9CYP2C19
SCHEMBL231888 0.86 ELANE (0.62) ELANECYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2385945-B1 TRIAZOLO AND TETRAZOLO PYRIMIDINE DERIVATIVES AS HNE INHIBITORS FOR TREATING COPD BAYER IP GMBH (DE) 2013-01-23 EP disclosed
WO-2010078953-A1 TRIAZOLO AND TETRAZOLO PYRIMIDINE DERIVATIVES AS HNE INHIBITORS FOR TREATING COPD BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-07-15 WO disclosed