SCHEMBL7904659

SCHEMBL7904659

COc1ccc(Cn2cncn2)cc1-c1cccc(NO)c1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 11/20 0.47
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
PDE4B Q07343 5/20 0.44
STS P08842 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3810121 0.84 PDE4B (0.52) CYP19A1PDE4BSTS
SCHEMBL8064800 0.84 HTT (0.52) HDAC1HDAC6PDE4B
SCHEMBL3805932 0.84 PDE4B (0.58) CYP19A1PDE4BSTS
SCHEMBL8067067 0.84 CYP19A1 (0.50) CYP19A1PDE4BSTS
SCHEMBL3805833 0.83 HDAC1 (0.51) CYP19A1HDAC1HDAC6STS
SCHEMBL4322642 0.83 CYP19A1 (0.55) CYP19A1HDAC1HDAC6PDE4BSTS
SCHEMBL4330785 0.82 HDAC1 (0.49) CYP19A1HDAC1HDAC6STS
SCHEMBL4322192 0.82 CYP19A1 (0.48) CYP19A1PDE4BSTS
SCHEMBL4323206 0.81 CYP19A1 (0.49) CYP19A1PDE4BSTS
SCHEMBL3809178 0.81 CYP19A1 (0.57) CYP19A1STS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059838-A2 PDE4 INHIBITORS SELECTIVE FOR THE LONG FORM OF PDE4 FOR TREATING INFLAMMATION AND AVOIDING SIDE EFFECTS DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed
WO-2009067600-A2 BIARYL PDE4 INHIBITORS FOR TREATING INFLAMMATION DECODE GENETICS EHF (IS) 2009-05-28 WO disclosed