SCHEMBL7904974

SCHEMBL7904974

CCCCCC(O)C(OC)c1cccc2c(=O)[nH]c(-c3cc(S(=O)(=O)N4CCOCC4)ccc3OCCC)nc12

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 20/20 0.56
PDE6C P51160 2/20 0.47
PDE6D O43924 1/20 0.47
PDE6A P16499 1/20 0.47
PDE6G P18545 1/20 0.47
PDE6B P35913 1/20 0.47
PDE6H Q13956 1/20 0.47
PDE11A Q9HCR9 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7902715 0.82 PDE5A (0.59) PDE5APDE6CPDE6DPDE6APDE6G
SCHEMBL7904959 0.82 PDE5A (0.69) PDE5APDE6CPDE6DPDE6APDE6G
SCHEMBL7899630 0.81 PDE5A (0.58) PDE5APDE6CPDE6DPDE6APDE6G
SCHEMBL7902825 0.81 PDE5A (0.48) PDE5APDE6CPDE6DPDE6APDE6G
SCHEMBL7901281 0.81 PDE5A (0.57) PDE5APDE6CPDE11A
SCHEMBL8672540 0.81 PDE5A (0.48) PDE5APDE6CPDE6DPDE6APDE6G
SCHEMBL7904851 0.80 PDE5A (0.58) PDE5APDE6CPDE6DPDE6APDE6G
SCHEMBL8140675 0.76 PDE5A (0.59) PDE5APDE6CPDE6DPDE6APDE6G
SCHEMBL7901187 0.76 PDE5A (0.55) PDE5APDE6CPDE11A
SCHEMBL8471415 0.75 PDE5A (0.62) PDE5APDE6CPDE6DPDE6APDE6G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187779-B1 ADMINISTERING ANTITUMOR AGENTS TO TREAT COLON CANCER CELL PATHWAYS, INC. 2001-02-13 US disclosed
US-5721238-A ANTIINFLAMMATORY AGENTS, CARDIOVASCULAR DISORDERS BAYER AKTIENGESELLSCHAFT (DE) 1998-02-24 US disclosed
EP-0722937-A1 2,8-Disubstituted quinazolinone BAYER AG (DE) 1996-07-24 EP disclosed