SCHEMBL790518

SCHEMBL790518

Cc1ccc(-c2ccccc2)c(F)c1O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.50
ELANE P08246 2/20 0.42
BACE1 P56817 2/20 0.41
ALOX5 P09917 1/20 0.41
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
BCL2L1 Q07817 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HDAC4 P56524 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
CYP2A6 P11509 1/20 0.39
CYP2B6 P20813 1/20 0.39
ALOX5AP P20292 1/20 0.38
FEN1 P39748 1/20 0.38
PTGS1 P23219 3/20 0.37
MEN1 O00255 2/20 0.37
PTGS2 P35354 2/20 0.37
KMT2A Q03164 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8459772 0.81 ESR2 (0.45) ESR2BACE1ALOX5ALDH1A1HPGD
SCHEMBL10617137 0.81 ESR2 (0.55) ESR2ELANEBACE1ALOX5ALDH1A1
Methane SCHEMBL28025030 0.79 ESR2 (0.53) ESR2ELANEBACE1ALOX5ALDH1A1
SCHEMBL1513737 0.79 ESR2 (0.53) ESR2ELANEBACE1ALOX5ALDH1A1
Ammonia Solution, Strong SCHEMBL27687172 0.79 ESR2 (0.44) ESR2BACE1ALOX5ALDH1A1HPGD
Methane SCHEMBL27747305 0.79 ESR2 (0.44) ESR2BACE1ALOX5ALDH1A1HPGD
SCHEMBL15861964 0.79 AKR1C3 (0.52) ALDH1A1AKR1C3AKR1C2
SCHEMBL25954438 0.78 ESR2 (0.42) ESR2ALDH1A1CYP2A6CYP2B6ALOX5AP
SCHEMBL15856373 0.78 ESR2 (0.42) ESR2ALDH1A1HSD17B10CYP2A6CYP2B6
SCHEMBL23789229 0.76 ESR2 (0.41) ESR2ALDH1A1CYP2A6CYP2B6ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2615918-A1 FATTY ACID SYNTHASE INHIBITORS GlaxoSmithKline Intellectual Property Development Limited (GB) 2013-07-24 EP disclosed
WO-2012037298-A1 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed