SCHEMBL7905308

SCHEMBL7905308

O=Cc1ccc(-c2ccc(-c3ccccc3)cc2)s1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.68
CYP2E1 P05181 2/20 0.61
CYP3A4 P08684 2/20 0.61
CYP2A6 P11509 2/20 0.61
CYP2C9 P11712 2/20 0.61
CYP2B6 P20813 2/20 0.61
CYP2C19 P33261 2/20 0.61
POLB P06746 2/20 0.52
RAB9A P51151 2/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
DPP4 P27487 1/20 0.50
PRF1 P14222 1/20 0.49
MAPT P10636 2/20 0.46
TDP1 Q9NUW8 1/20 0.45
KDM4E B2RXH2 2/20 0.44
HPGD P15428 2/20 0.44
GAA P10253 1/20 0.44
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL70783 0.96 APP (0.67) APPCYP2E1CYP3A4CYP2A6CYP2C9
SCHEMBL10472980 0.92 APP (0.73) APPCYP2E1CYP3A4CYP2A6CYP2C9
SCHEMBL7006689 0.86 APP (0.91) APPCYP2E1CYP3A4CYP2A6CYP2C9
SCHEMBL28831708 0.84 APP (0.59) APPCYP2E1CYP3A4CYP2A6CYP2C9
SCHEMBL30903820 0.84 APP (0.94) APPCYP2E1CYP3A4CYP2A6CYP2C9
SCHEMBL5399485 0.84 APP (0.94) APPCYP2E1CYP3A4CYP2A6CYP2C9
SCHEMBL30903823 0.84 APP (0.94) APPCYP2E1CYP3A4CYP2A6CYP2C9
SCHEMBL30903822 0.84 APP (0.94) APPCYP2E1CYP3A4CYP2A6CYP2C9
SCHEMBL14713496 0.81 APP (1.00) APPCYP2E1CYP3A4CYP2A6CYP2C9
SCHEMBL2592315 0.81 APP (1.00) APPCYP2E1CYP3A4CYP2A6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015172047-A1 CYCLIC PEPTIDE COMPOUNDS AND RELATED METHODS, SALTS AND COMPOSITIONS MERCK SHARP & DOHME CORP. (US) 2015-11-12 WO disclosed
WO-2010075215-A1 NOVEL ANTIBACTERIAL AGENTS FOR THE TREATMENT OF GRAM POSITIVE INFECTIONS CUBIST PHARMACEUTICALS, INC. (US) 2010-07-01 WO disclosed