SCHEMBL790547

SCHEMBL790547

O=C1OCCC1(F)COCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 5/20 0.41
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
LMNA P02545 1/20 0.37
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
MMP9 P14780 1/20 0.36
GRM5 P41594 2/20 0.36
OPRM1 P35372 1/20 0.35
KCNH2 Q12809 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
MAOB P27338 3/20 0.34
DAO P14920 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
NFKB1 P19838 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25131500 0.79 TACR1 (0.41) TACR1TSHRNPSR1MEN1KMT2A
SCHEMBL25131487 0.77 TACR1 (0.40) TACR1TSHRNPSR1MEN1KMT2A
SCHEMBL20512123 0.74 TACR1 (0.40) TACR1TSHRNPSR1MEN1KMT2A
SCHEMBL27674725 0.73 TSHR (0.47) TACR1TSHRNPSR1MEN1KMT2A
SCHEMBL28306256 0.72 TSHR (0.54) TACR1TSHRSLC6A4
SCHEMBL25131484 0.71 MAPT (0.36) TACR1TSHRNPSR1MAOBALDH1A1
SCHEMBL599239 0.70 TSHR (0.47) TACR1TSHRLMNAMMP2MMP3
Oxirane SCHEMBL3317346 0.69 TSHR (0.75) TACR1TSHRNPSR1MEN1KMT2A
SCHEMBL15105750 0.69 TACR1 (0.46) TACR1TSHRKMT2AGRM5ALDH1A1
SCHEMBL2221074 0.68 TSHR (0.48) TACR1TSHRNPSR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616080-A1 2' -FLUORO SUBSTITUTED CARBA-NUCLEOSIDE ANALOGS FOR ANTIVIRAL TREATMENT Gilead Sciences, Inc. (US) 2013-07-24 EP disclosed
WO-2012037038-A1 2' -FLUORO SUBSTITUTED CARBA-NUCLEOSIDE ANALOGS FOR ANTIVIRAL TREATMENT GILEAD SCIENCES, INC. (US) 2012-03-22 WO disclosed