SCHEMBL7905620

SCHEMBL7905620

CCOC(=O)c1cc(CBr)cc(COCCOC)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.46
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
CA7 P43166 3/20 0.46
CA9 Q16790 3/20 0.46
CA14 Q9ULX7 3/20 0.46
CYP4F2 P78329 2/20 0.41
CYP4A11 Q02928 2/20 0.41
HSD17B2 P37059 1/20 0.40
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
KMT2A Q03164 5/20 0.39
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 3/20 0.39
TSHR P16473 2/20 0.39
PTGER4 P35408 2/20 0.39
MAPT P10636 2/20 0.39
ABCB11 O95342 1/20 0.39
CYP3A4 P08684 1/20 0.39
ADRA2B P18089 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7592102 0.84 CA12 (0.58) CA12CA1CA2CA7CA9
SCHEMBL7594237 0.83 PKM (0.38) CA12CA1CA2CA7CA9
SCHEMBL9885271 0.81 CA12 (0.55) CA12CA1CA2CA7CA9
SCHEMBL2212198 0.81 CA12 (0.58) CA12CA1CA2CA7CA9
SCHEMBL9886090 0.80 CA12 (0.51) CA12CA1CA2CA7CA9
SCHEMBL7595272 0.80 MEN1 (0.43) CA12CA1CA2CA7CA9
SCHEMBL16528056 0.76 CA12 (0.53) CA12CA1CA2CA7CA9
SCHEMBL4652540 0.75 CYP2C19 (0.57) CA12CA1CA2CA7CA9
SCHEMBL7896250 0.75 MAPT (0.48) CA12CA1CA2CA7CA9
SCHEMBL13307487 0.74 CA12 (0.50) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6200981-B1 FOR TREATING INFLAMMATORY DISEASES SUCH AS ASTHMA, INFLAMMATORY BOWEL DISEASE, PSORIASIS, RHEUMATOID ARTHRITIS, MYOCARDIAL ISCHAEMIA, CYSTIC FIBROSIS, ARTHEREOSCLEROSIS, RESTENOSIS, PERIDONTAL DISEASE, SEPTIC SHOCK, OSTEOARTHRITIS ASTRAZENECA UK LIMITED (GB) 2001-03-13 US disclosed