SCHEMBL7905978

SCHEMBL7905978

Nc1cccc(-c2cccc(O)n2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.53
MEN1 O00255 4/20 0.53
KDM4E B2RXH2 3/20 0.53
MAPT P10636 3/20 0.53
KMT2A Q03164 3/20 0.53
LMNA P02545 3/20 0.53
HPGD P15428 2/20 0.53
PLK1 P53350 1/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
TSHR P16473 1/20 0.49
RECQL P46063 1/20 0.49
GLA P06280 1/20 0.49
METAP2 P50579 1/20 0.47
MAOA P21397 1/20 0.47
KARS1 Q15046 1/20 0.46
MAP4K4 O95819 2/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1028576 0.77 MEN1 (0.68) ALDH1A1MEN1MAPTKMT2AHPGD
SCHEMBL1040984 0.77 TSHR (0.57) ALDH1A1MEN1KDM4EMAPTKMT2A
SCHEMBL7086276 0.74 MEN1 (0.39) ALDH1A1MEN1KDM4EMAPTKMT2A
SCHEMBL11804494 0.74 MAP4K4 (0.54) ALDH1A1MEN1KDM4EMAPTKMT2A
SCHEMBL1074467 0.73 ALDH1A1 (0.46) ALDH1A1MEN1KDM4EMAPTKMT2A
SCHEMBL17174081 0.73 MEN1 (0.53) ALDH1A1MEN1KDM4EMAPTKMT2A
SCHEMBL11182648 0.73 TSHR (0.53) ALDH1A1MEN1KDM4EMAPTKMT2A
SCHEMBL2627239 0.73 NPC1 (0.49) ALDH1A1MEN1KDM4EMAPTKMT2A
SCHEMBL13040762 0.73 IDO1 (0.51) ALDH1A1MEN1MAPTKMT2AHPGD
SCHEMBL27646975 0.73 TSHR (0.66) ALDH1A1MEN1KDM4EMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211220-B1 ANTITUMOR AGENTS AND ANTICARCIINOGENIC AGENTS CELL PATHWAYS, INC. 2001-04-03 US disclosed
WO-1994029277-A1 AMILINO- OR PYRIDYLAMINO- CYCLOBUTENE- 1,2-DIONE DERIVATIVES AS cGMP PHOSPHODIESTERASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1994-12-22 WO disclosed