SCHEMBL7906040

SCHEMBL7906040

O=NCc1cccc2c1Cc1c-2[nH]c(=O)c2c1CCCC2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ALOX15 P16050 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD11B1 P28845 2/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
BRD4 O60885 3/20 0.32
CCNB2 O95067 1/20 0.32
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32
GSK3B P49841 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
CCNB3 Q8WWL7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13086601 0.85 CCNB2 (0.41) HPGDKDM4EALDH1A1TSHRHSD17B10
SCHEMBL7897594 0.84 HPGD (0.36) HPGDKDM4EALDH1A1TSHRHSD17B10
SCHEMBL3057285 0.84 PNMT (0.43) HPGDKDM4EALDH1A1TSHRHSD17B10
SCHEMBL2790481 0.84 CHEK1 (0.43) HPGDKDM4EALDH1A1TSHRHSD17B10
SCHEMBL3045256 0.81 PARP1 (0.38) HPGDKDM4EALDH1A1TSHRHSD17B10
SCHEMBL3066815 0.80 KDR (0.42) HPGDKDM4EALDH1A1HSD17B10
SCHEMBL7897601 0.79 BRD4 (0.36) HPGDKDM4EALDH1A1TSHRHSD17B10
SCHEMBL2782051 0.79 KDR (0.41) HPGDKDM4EALDH1A1HSD17B10
SCHEMBL3054827 0.79 PARP1 (0.39) HPGDKDM4EALDH1A1TSHRHSD17B10
SCHEMBL2780726 0.79 KDR (0.41) HPGDKDM4EALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010077663-A2 SUBSTITUTED TETRACYCLIC 1H-INDENO (1,2-B) PYRIDINE-2 (5H)-ONE ANALOGS THEREOF AND USES THEREOF INOTEK PHARMACEUTICALS CORPORATION (US) 2010-07-08 WO disclosed