SCHEMBL7907906

SCHEMBL7907906

O=C(O)CN1C(=O)C(NC(=O)c2ccccc2)CN(C(=O)CCc2ccccc2)c2ccccc21

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 2/20 0.71
CYP3A4 P08684 4/20 0.52
XIAP P98170 4/20 0.52
ACE P12821 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3063918 1.00 CASP1 (0.71) CASP1CYP3A4XIAPACE
SCHEMBL644745 0.90 CASP1 (0.67) CASP1CYP3A4XIAP
SCHEMBL12831227 0.90 CASP1 (0.72) CASP1CYP3A4XIAP
SCHEMBL645652 0.90 CASP1 (0.60) CASP1CYP3A4XIAPACE
SCHEMBL645651 0.90 CASP1 (0.60) CASP1CYP3A4XIAPACE
SCHEMBL12994842 0.87 CASP1 (0.65) CASP1CYP3A4XIAP
SCHEMBL10284729 0.85 CASP1 (0.60) CASP1CYP3A4XIAP
SCHEMBL646012 0.85 CASP1 (0.63) CASP1CYP3A4XIAP
SCHEMBL646010 0.85 CASP1 (0.63) CASP1CYP3A4XIAP
SCHEMBL12994889 0.84 CASP1 (0.64) CASP1CYP3A4XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6204261-B1 Inhibitors of interleukin-1β Converting enzyme inhibitors VERTEX PHARMACEUTICALS INCORPORATED 2001-03-20 US disclosed