SCHEMBL7909506

SCHEMBL7909506

CCCCC[C@H](C#N)c1ccccc1C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.37
CYP3A4 P08684 3/20 0.37
CYP2C9 P11712 3/20 0.37
TSHR P16473 3/20 0.37
CYP2C19 P33261 3/20 0.37
AR P10275 3/20 0.35
CTSK P43235 1/20 0.35
MC4R P32245 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TP53 P04637 1/20 0.34
HSD11B1 P28845 2/20 0.34
TLR8 Q9NR97 1/20 0.34
SLC6A4 P31645 1/20 0.33
ACP3 P15309 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CNR2 P34972 1/20 0.33
KCNH2 Q12809 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28776287 0.89 CTSK (0.37) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL909422 0.85 CCR1 (0.35) ARMC4RHSD11B1SLC6A4ACP3
SCHEMBL3695512 0.85 CCR1 (0.35) ARMC4RHSD11B1SLC6A4ACP3
SCHEMBL720614 0.80 ACP3 (0.39) ARMC4RSMN1; SMN2SLC6A4ACP3
SCHEMBL194438 0.80 ACP3 (0.36) ARMC4RHSD11B1SLC6A4ACP3
SCHEMBL23169003 0.80 CYSLTR2 (0.41) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL19292942 0.78 CYSLTR2 (0.40) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL9232277 0.78 CYP1A2 (0.39) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL31036078 0.78 ESR1 (0.36) TSHRMAPTCNR2P2RX7
SCHEMBL16442414 0.78 CYP1A2 (0.39) CYP1A2CYP3A4CYP2C9TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010098496-A1 PROCESS FOR PRODUCING TETRAHYDROTRIAZOLOPYRIDINE DERIVATIVE EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-09-02 WO disclosed