SCHEMBL7909698

SCHEMBL7909698

c1ccc(COc2ccc(Nc3ncnc4cnc(-c5ccc(CN6CCCCC6)o5)cc34)cc2)cc1

nearest known ligand 0.75

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 14/20 0.75
EGFR P00533 12/20 0.70
ERBB4 Q15303 2/20 0.50
CHEK2 O96017 1/20 0.50
ROS1 P08922 1/20 0.50
FLT3 P36888 1/20 0.50
AURKB Q96GD4 1/20 0.50
CLK4 Q9HAZ1 1/20 0.50
MKNK2 Q9HBH9 1/20 0.50
JAK3 P52333 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4559023 0.92 ERBB2 (0.72) ERBB2EGFRERBB4CHEK2ROS1
SCHEMBL27518939 0.88 ERBB2 (0.78) ERBB2EGFRERBB4CHEK2ROS1
SCHEMBL7005564 0.86 ERBB2 (1.00) ERBB2EGFRERBB4CHEK2ROS1
Hydrochloric Acid SCHEMBL7013332 0.85 ERBB2 (0.98) ERBB2EGFRERBB4CHEK2ROS1
SCHEMBL4359057 0.83 ERBB2 (0.79) ERBB2EGFRERBB4CHEK2ROS1
SCHEMBL7009350 0.83 ERBB2 (0.66) ERBB2EGFRERBB4
SCHEMBL7006741 0.83 ERBB2 (0.66) ERBB2EGFRERBB4
Hydrochloric Acid SCHEMBL7007235 0.83 ERBB2 (0.65) ERBB2EGFR
Dimethylamine SCHEMBL7099762 0.83 ERBB2 (0.65) ERBB2EGFRERBB4CHEK2ROS1
Hydrochloric Acid SCHEMBL7915742 0.83 ERBB2 (0.65) ERBB2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6207669-B1 IN TREATMENT OF CANCER AND PSORIASIS GLAXO WELLCOME INC. 2001-03-27 US disclosed