SCHEMBL4359057

SCHEMBL4359057

CN(C)Cc1ccc(-c2cc3c(Nc4ccc(OCc5ccccc5)cc4)ncnc3cn2)o1

nearest known ligand 0.79

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 15/20 0.79
EGFR P00533 13/20 0.70
AURKB Q96GD4 2/20 0.53
ERBB4 Q15303 2/20 0.53
CHEK2 O96017 1/20 0.53
ROS1 P08922 1/20 0.53
FLT3 P36888 1/20 0.53
CLK4 Q9HAZ1 1/20 0.53
MKNK2 Q9HBH9 1/20 0.53
TTBK1 Q5TCY1 1/20 0.46
TTBK2 Q6IQ55 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7005564 0.89 ERBB2 (1.00) ERBB2EGFRAURKBERBB4CHEK2
SCHEMBL7010246 0.88 ERBB2 (0.72) ERBB2EGFRAURKBERBB4CHEK2
Hydrochloric Acid SCHEMBL7013332 0.88 ERBB2 (0.98) ERBB2EGFRAURKBERBB4CHEK2
SCHEMBL7007882 0.88 ERBB2 (0.76) ERBB2EGFR
SCHEMBL27518939 0.85 ERBB2 (0.78) ERBB2EGFRAURKBERBB4CHEK2
SCHEMBL4559023 0.84 ERBB2 (0.72) ERBB2EGFRAURKBERBB4CHEK2
SCHEMBL7909698 0.83 ERBB2 (0.75) ERBB2EGFRAURKBERBB4CHEK2
SCHEMBL7005311 0.83 ERBB2 (1.00) ERBB2EGFRAURKBERBB4CHEK2
SCHEMBL7890178 0.83 ERBB2 (0.77) ERBB2EGFRAURKBERBB4CHEK2
SCHEMBL7007362 0.83 ERBB2 (1.00) ERBB2EGFRAURKBERBB4CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1230185-A Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors GLAXO GROUP LTD (GB) 1999-09-29 CN claimed
WO-2009070328-A1 MODULATORS OF THE EPIDERMAL GROWTH FACTOR RECEPTOR (EGFR) PATHWAY FOR USE IN THE TREATMENT OR PREVENTION OF SUBSTANCE ABUSE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2009-06-04 WO disclosed