SCHEMBL7910364

SCHEMBL7910364

Cc1nc(-c2ccc(C(=O)N3CCC(C(=O)NC(C4=CC=C(F)CC4)C(F)(F)F)(c4ccc(F)cc4)CC3)cc2)no1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 10/20 0.39
HDAC6 Q9UBN7 2/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
TACR3 P29371 2/20 0.38
GRM5 P41594 1/20 0.38
CLPP Q16740 1/20 0.38
MGLL Q99685 1/20 0.37
STAT3 P40763 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
PLK1 P53350 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7909985 0.91 TACR3 (0.39) HDAC4HDAC6HDAC2HDAC8TACR3
SCHEMBL7915785 0.89 TACR3 (0.40) HDAC4HDAC6HDAC2HDAC8TACR3
SCHEMBL13092384 0.89 HDAC4 (0.42) HDAC4HDAC6HDAC2HDAC8TACR3
SCHEMBL7912369 0.83 TACR3 (0.40) HDAC4HDAC6HDAC2HDAC8TACR3
SCHEMBL13092395 0.82 TACR3 (0.42) HDAC4HDAC6HDAC2HDAC8TACR3
SCHEMBL7909169 0.82 TACR3 (0.41) HDAC4HDAC6HDAC2HDAC8TACR3
SCHEMBL13092382 0.81 TACR3 (0.41) HDAC4HDAC6HDAC2HDAC8TACR3
SCHEMBL13092381 0.80 TACR3 (0.44) HDAC4HDAC6HDAC2HDAC8TACR3
SCHEMBL378447 0.79 MGLL (0.48) HDAC4HDAC6HDAC2HDAC8TACR3
SCHEMBL13092247 0.79 MGLL (0.44) HDAC4HDAC6HDAC2HDAC8TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010106081-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-23 WO disclosed