SCHEMBL7911458

SCHEMBL7911458

Cc1c(C(=O)N[C@@H](O)c2cccc(F)c2)c2cccc(F)c2c(=O)n1Cc1cccs1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 1/20 0.40
KLK1 P06870 1/20 0.40
CNR2 P34972 1/20 0.39
RAB9A P51151 8/20 0.38
NPC1 O15118 6/20 0.38
MAPK1 P28482 2/20 0.37
MAPT P10636 8/20 0.37
LMNA P02545 5/20 0.37
TSHR P16473 4/20 0.37
TP53 P04637 3/20 0.37
ALDH1A1 P00352 4/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.35
RECQL P46063 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HTT P42858 2/20 0.34
USP2 O75604 1/20 0.34
ESR1 P03372 1/20 0.34
GNRHR P30968 2/20 0.34
KDM4E B2RXH2 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1366825 0.88 CYP2C9 (0.46) KLKB1KLK1CNR2RAB9ANPC1
SCHEMBL7918066 0.85 PPARG (0.39) CNR2MAPTTP53ALDH1A1GNRHR
SCHEMBL7914678 0.85 POLB (0.36) TP53ALDH1A1SMN1; SMN2RECQLGNRHR
SCHEMBL7914357 0.84 TP53 (0.40) MAPTTP53GNRHRPOLB
SCHEMBL7914360 0.83 S1PR3 (0.39) L3MBTL1
SCHEMBL12151037 0.83 S1PR3 (0.37) TP53GNRHRPOLB
SCHEMBL11920290 0.82 GNRHR (0.36) CNR2LMNASMN1; SMN2GNRHR
SCHEMBL11920581 0.82 GNRHR (0.39) CNR2GNRHR
SCHEMBL7911647 0.82 GNRHR (0.42) MAPK1LMNATP53GNRHRPOLB
SCHEMBL7914022 0.81 ROCK2 (0.33) MAPK1TP53GNRHRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010045948-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-04-29 WO disclosed