SCHEMBL7913161

SCHEMBL7913161

c1cncc(P(CCP(c2cccnc2)c2cccnc2)c2cccnc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.44
CYP1A2 P05177 3/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 2/20 0.40
CHRNA7 P36544 1/20 0.39
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CHRNB2 P17787 2/20 0.38
CHRNA4 P43681 2/20 0.38
HRH4 Q9H3N8 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
THRB P10828 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30480022 0.81 CYP11B1 (0.35) CYP2A6CYP1A2ALDH1A1CYP3A4CYP2D6
SCHEMBL30319508 0.77 ALDH1A1 (0.50) CYP2A6CYP1A2ALDH1A1CYP3A4CYP2D6
SCHEMBL617000 0.77 ALDH1A1 (0.50) CYP2A6CYP1A2ALDH1A1CYP3A4CYP2D6
SCHEMBL15652709 0.75 ALDH1A1 (0.48) CYP2A6CYP1A2ALDH1A1CYP3A4CYP2D6
SCHEMBL29143382 0.73
SCHEMBL12620100 0.73
SCHEMBL7919893 0.72 KCNA5 (0.42) CYP1A2ALDH1A1CYP3A4CYP2D6MAPT
SCHEMBL617213 0.71 CYP3A4 (0.57) CYP2A6CYP1A2ALDH1A1CYP3A4KDM4E
SCHEMBL4833637 0.71 ALDH1A1 (0.44) CYP2A6CYP1A2ALDH1A1CYP3A4CYP2D6
SCHEMBL4833644 0.71 CYP2A6 (0.44) CYP2A6CYP1A2ALDH1A1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6218378-B1 FOR THERAPY OR INHIBITION OF OVARIAN TUMORS, CERVICAL TUMORS, LUNG CANCER AND MELANOMA GRIFFITH UNIVERSITY (AU) 2001-04-17 US disclosed
US-6159957-A Method of treatment or inhibition of tumors using pyridyl-substituted metal-diphosphine complexes GRIFFITH UNIVERSITY (AU) 2000-12-12 US disclosed