SCHEMBL7914640

SCHEMBL7914640

COc1ccc(Cc2ccc(OC)c(-c3cccc(Cl)c3)c2F)cn1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.45
EPHB4 P54760 1/20 0.45
TEK Q02763 1/20 0.45
PDE4B Q07343 7/20 0.40
PDE4D Q08499 3/20 0.40
CYP2C9 P11712 1/20 0.40
GRM2 Q14416 1/20 0.39
FYN P06241 1/20 0.36
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
HCRTR1 O43613 2/20 0.35
HCRTR2 O43614 2/20 0.35
CTSA P10619 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4325092 0.91 PDE4B (0.39) KDREPHB4TEKPDE4BPDE4D
SCHEMBL3467239 0.90 PDE4B (0.41) PDE4BPDE4DFYNNPC1MAPT
SCHEMBL8067934 0.89 PDE4B (0.41) PDE4BPDE4DNPC1MAPTTSHR
SCHEMBL3795717 0.89 HTR1A (0.38) KDREPHB4TEKPDE4BPDE4D
SCHEMBL3467151 0.88 PDE4B (0.39) PDE4BPDE4DFYNNPC1MAPT
SCHEMBL7902765 0.88 PDE4B (0.39) PDE4BPDE4DFYNHCRTR1HCRTR2
SCHEMBL8024594 0.88 PDE4B (0.42) PDE4BPDE4DFYNNPC1MAPT
SCHEMBL4323960 0.88 PDE4B (0.41) PDE4BPDE4DMAPT
SCHEMBL3468023 0.87 PDE4B (0.42) PDE4BPDE4DFYN
SCHEMBL3798675 0.87 PDE4B (0.42) PDE4BPDE4DGRM2FYNNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059838-A2 PDE4 INHIBITORS SELECTIVE FOR THE LONG FORM OF PDE4 FOR TREATING INFLAMMATION AND AVOIDING SIDE EFFECTS DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed