SCHEMBL7914942

SCHEMBL7914942

Nc1cccc(-n2ccc(=O)c(-c3ccnn3-c3ccnc4ccccc34)n2)c1

nearest known ligand 0.74

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 6/20 0.74
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HTT P42858 1/20 0.35
PKM P14618 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33
GRM4 Q14833 1/20 0.33
KCNH2 Q12809 1/20 0.32
AR P10275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2501874 0.87 PDE10A (0.71) PDE10AALDH1A1
SCHEMBL2750597 0.86 PDE10A (0.70) PDE10AALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL2472403 0.86 PDE10A (0.70) PDE10AALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL3506103 0.85 PDE10A (0.78) PDE10AALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL3504464 0.85 PDE10A (0.78) PDE10AALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL3505967 0.85 PDE10A (1.00) PDE10AALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL2503777 0.84 PDE10A (0.73) PDE10AALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL2480986 0.83 PDE10A (0.66) PDE10AALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL7911573 0.83 PDE10A (0.65) PDE10AALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL7911641 0.82 PDE10A (0.68) PDE10AALDH1A1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063610-A1 PYRIDAZINONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-06-10 WO disclosed