SCHEMBL7915547

SCHEMBL7915547

NC1=N[C@@]2(c3cc(-c4cccnc4F)ccc3F)COCCC2CS1

nearest known ligand 0.64

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.64
CTSD P07339 3/20 0.56
CYP2D6 P10635 1/20 0.50
KCNH2 Q12809 1/20 0.50
CTSB P07858 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3295791 1.00 BACE1 (0.64) BACE1CTSDCYP2D6KCNH2CTSB
SCHEMBL3295793 1.00 BACE1 (0.64) BACE1CTSDCYP2D6KCNH2CTSB
SCHEMBL8023214 0.86 BACE1 (0.53) BACE1CTSDCTSB
SCHEMBL2620242 0.86 BACE1 (0.53) BACE1CTSDCTSB
SCHEMBL2933567 0.86 BACE1 (0.53) BACE1CTSDCTSB
SCHEMBL7922748 0.83 BACE1 (0.55) BACE1CTSDKCNH2CTSB
SCHEMBL3302100 0.83 BACE1 (0.55) BACE1CTSDKCNH2CTSB
SCHEMBL2341633 0.83 BACE1 (0.55) BACE1CTSDKCNH2CTSB
SCHEMBL1935618 0.83 BACE1 (0.67) BACE1CTSDCYP2D6KCNH2
SCHEMBL3300779 0.82 BACE1 (0.52) BACE1CTSDCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038686-A1 NOVEL FUSED AMINODIHYDROTHIAZINE DERIVATIVE エーザイ・アール・アンド・ディー・マネジメント株式会社 (JP) 2010-04-08 WO disclosed