SCHEMBL7922748

SCHEMBL7922748

NC1=NC2(c3cc(-c4cccnc4F)cs3)COCC[C@H]2CS1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.55
KCNH2 Q12809 1/20 0.49
CTSD P07339 3/20 0.47
CTSB P07858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3302100 1.00 BACE1 (0.55) BACE1KCNH2CTSDCTSB
SCHEMBL2341633 1.00 BACE1 (0.55) BACE1KCNH2CTSDCTSB
SCHEMBL2620310 0.85 BACE1 (0.47) BACE1CTSDCTSB
SCHEMBL2927948 0.85 BACE1 (0.47) BACE1CTSDCTSB
SCHEMBL7915547 0.83 BACE1 (0.64) BACE1KCNH2CTSDCTSB
SCHEMBL3295791 0.83 BACE1 (0.64) BACE1KCNH2CTSDCTSB
SCHEMBL3295793 0.83 BACE1 (0.64) BACE1KCNH2CTSDCTSB
SCHEMBL7927114 0.77 BACE1 (0.59) BACE1KCNH2
SCHEMBL3299449 0.77 BACE1 (0.59) BACE1KCNH2
SCHEMBL9913157 0.77 BACE1 (0.59) BACE1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038686-A1 NOVEL FUSED AMINODIHYDROTHIAZINE DERIVATIVE エーザイ・アール・アンド・ディー・マネジメント株式会社 (JP) 2010-04-08 WO disclosed