SCHEMBL7916643

SCHEMBL7916643

COC[C@H]1CC2CSC(N)=NC2(c2cc(C(C)=O)ccc2F)CO1

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.72
BACE2 Q9Y5Z0 2/20 0.68
CTSD P07339 1/20 0.54
KCNH2 Q12809 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3305419 0.86 BACE1 (0.54) BACE1BACE2CTSDKCNH2
SCHEMBL7916622 0.85 BACE1 (0.77) BACE1BACE2CTSD
SCHEMBL7918277 0.84 BACE1 (1.00) BACE1BACE2CTSD
SCHEMBL9913117 0.84 BACE1 (1.00) BACE1BACE2CTSD
SCHEMBL9913118 0.83 BACE1 (0.71) BACE1BACE2CTSD
SCHEMBL2342407 0.83 BACE1 (0.50) BACE1BACE2CTSDKCNH2
SCHEMBL7927883 0.83 BACE1 (0.50) BACE1BACE2CTSDKCNH2
SCHEMBL3300713 0.82 BACE1 (0.79) BACE1BACE2KCNH2
SCHEMBL3300708 0.82 BACE1 (0.79) BACE1BACE2KCNH2
SCHEMBL15630354 0.81 BACE1 (1.00) BACE1BACE2CTSDKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038686-A1 NOVEL FUSED AMINODIHYDROTHIAZINE DERIVATIVE エーザイ・アール・アンド・ディー・マネジメント株式会社 (JP) 2010-04-08 WO disclosed