SCHEMBL7917241

SCHEMBL7917241

CCCOc1cc2c(c3c(=O)c(-c4ccc(OC)cc4)cn(COP(=O)(O)OC)c13)OCC2

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.33
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
CLK1 P49759 1/20 0.31
RAB9A P51151 1/20 0.31
PDE4B Q07343 1/20 0.30
TYMS P04818 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7907760 0.94 ABCB1 (0.34) ABCB1CNR1CNR2ESR1ESR2
SCHEMBL2578934 0.89 ABCB1 (0.33) ABCB1CNR1CNR2ESR1ESR2
SCHEMBL12160480 0.88 ABCB1 (0.31) ABCB1
SCHEMBL2584574 0.86 ABCB1 (0.32) ABCB1CNR1CNR2
SCHEMBL12160478 0.85 ESR1 (0.38) ABCB1CNR1CNR2ESR1ESR2
SCHEMBL7910534 0.84
SCHEMBL7912511 0.83 RAB9A (0.41) ABCB1CNR1CNR2ESR1ESR2
SCHEMBL2587899 0.83 ABCB1 (0.30) ABCB1
SCHEMBL12160475 0.83 BCHE (0.39) ESR1ESR2
SCHEMBL2586348 0.81 ESR1 (0.37) ABCB1CNR1CNR2ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010064735-A1 QUINOLONE COMPOUND AND PHARMACEUTICAL COMPOSITION OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2010-06-10 WO disclosed