SCHEMBL7917992

SCHEMBL7917992

COc1ccc(Cc2ccc(CNC(=O)N(C)C)nc2)c(F)c1-c1cccc(N)c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.38
GRM2 Q14416 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CTSA P10619 1/20 0.34
HCRTR1 O43613 3/20 0.33
HCRTR2 O43614 3/20 0.33
KIT P10721 1/20 0.33
WDR5 P61964 1/20 0.33
TP53 P04637 1/20 0.33
CHRM4 P08173 1/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
FFAR1 O14842 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8065009 0.90 HCRTR1 (0.39) CTSAHCRTR1HCRTR2WDR5
Hydrochloric Acid SCHEMBL4325701 0.89 HCRTR1 (0.39) MEN1KMT2ACYP1A2CYP2C19CTSA
SCHEMBL8072156 0.82 GRM2 (0.42) GRM2CTSAKITFFAR1
SCHEMBL8072151 0.82 CD274 (0.37) GRM2CTSAKITFFAR1
SCHEMBL3791157 0.81 PDE4D (0.45) ADORA2AMEN1KMT2ACYP1A2CYP2C19
SCHEMBL8070837 0.81 FFAR1 (0.39) GRM2CTSAKITFFAR1
SCHEMBL3792183 0.80 PDE4D (0.42) ADORA2AMEN1KMT2ACYP1A2CYP2C19
SCHEMBL8066309 0.80 MAP4K4 (0.42) KIT
SCHEMBL7916577 0.80 PDE4D (0.41) CTSAHCRTR1HCRTR2WDR5
SCHEMBL7913183 0.79 MAPK1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059838-A2 PDE4 INHIBITORS SELECTIVE FOR THE LONG FORM OF PDE4 FOR TREATING INFLAMMATION AND AVOIDING SIDE EFFECTS DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed