SCHEMBL7918276

SCHEMBL7918276

COC[C@H]1CC2CSC(NC(=O)c3ccccc3)=NC2(c2ccccc2F)CO1

nearest known ligand 0.66

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.66
BACE2 Q9Y5Z0 1/20 0.54
KCNH2 Q12809 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9913407 1.00 BACE1 (0.66) BACE1BACE2KCNH2
SCHEMBL17296552 0.90 BACE1 (0.53) BACE1BACE2KCNH2
SCHEMBL15783590 0.90 BACE1 (0.53) BACE1BACE2KCNH2
SCHEMBL17296556 0.88 BACE1 (0.65) BACE1BACE2KCNH2
SCHEMBL15783588 0.88 BACE1 (0.65) BACE1BACE2KCNH2
SCHEMBL7922737 0.86 BACE1 (0.67) BACE1BACE2KCNH2
SCHEMBL9913311 0.86 BACE1 (0.67) BACE1BACE2KCNH2
SCHEMBL14716731 0.83 BACE1 (0.72) BACE1BACE2
SCHEMBL15369962 0.82 BACE1 (0.61) BACE1BACE2
SCHEMBL15369963 0.82 BACE1 (0.64) BACE1BACE2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038686-A1 NOVEL FUSED AMINODIHYDROTHIAZINE DERIVATIVE エーザイ・アール・アンド・ディー・マネジメント株式会社 (JP) 2010-04-08 WO disclosed