SCHEMBL7918279

SCHEMBL7918279

COC[C@H]1CC2CSC(NC(=O)OC(C)(C)C)=N[C@@]2(c2cc([N+](=O)[O-])ccc2F)CO1

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.48
BACE2 Q9Y5Z0 3/20 0.46
KCNH2 Q12809 2/20 0.37
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9913116 1.00 BACE1 (0.48) BACE1BACE2KCNH2CYP2D6
SCHEMBL7925015 0.93 BACE1 (0.46) BACE1BACE2KCNH2CYP2D6
SCHEMBL9913148 0.93 BACE1 (0.45) BACE1BACE2KCNH2CYP2D6
SCHEMBL7922169 0.93 BACE1 (0.45) BACE1BACE2KCNH2CYP2D6
SCHEMBL2619867 0.90 DRD2 (0.36) BACE1BACE2KCNH2
SCHEMBL7924326 0.89 BACE1 (0.47) BACE1BACE2KCNH2CYP2D6
SCHEMBL9913107 0.89 BACE1 (0.47) BACE1BACE2KCNH2CYP2D6
SCHEMBL9913119 0.88 BACE1 (0.55) BACE1BACE2KCNH2CYP2D6
SCHEMBL7927020 0.88 BACE1 (0.55) BACE1BACE2KCNH2CYP2D6
SCHEMBL15171753 0.87 BACE1 (0.36) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038686-A1 NOVEL FUSED AMINODIHYDROTHIAZINE DERIVATIVE エーザイ・アール・アンド・ディー・マネジメント株式会社 (JP) 2010-04-08 WO disclosed