SCHEMBL7918892

SCHEMBL7918892

CC1COCC2(c3cc(N)ccc3F)N=C(NC(=O)OC(C)(C)C)SCC12

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 17/20 0.40
BACE2 Q9Y5Z0 14/20 0.40
CYP2D6 P10635 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2340636 1.00 BACE1 (0.40) BACE1BACE2CYP2D6KCNH2
SCHEMBL7927021 1.00 BACE1 (0.40) BACE1BACE2CYP2D6KCNH2
SCHEMBL9913131 1.00 BACE1 (0.40) BACE1BACE2CYP2D6KCNH2
SCHEMBL7924432 0.93 BACE1 (0.40) BACE1BACE2
SCHEMBL9913134 0.91 BACE1 (0.38) BACE1BACE2
SCHEMBL7922777 0.91 BACE1 (0.38) BACE1BACE2
SCHEMBL7928138 0.91 BACE1 (0.38) BACE1BACE2
SCHEMBL8031655 0.90 BACE1 (0.50) BACE1BACE2CYP2D6KCNH2
SCHEMBL8020348 0.90 BACE1 (0.50) BACE1BACE2CYP2D6KCNH2
SCHEMBL2619832 0.90 BACE1 (0.50) BACE1BACE2CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038686-A1 NOVEL FUSED AMINODIHYDROTHIAZINE DERIVATIVE エーザイ・アール・アンド・ディー・マネジメント株式会社 (JP) 2010-04-08 WO disclosed