SCHEMBL7920436

SCHEMBL7920436

COc1ccc(NC(=O)C2(c3noc(C)n3)C=CC(c3ccccc3C)=CC2)cc1OC[C@@H]1CCCN1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.43
CHRNB4 P30926 4/20 0.41
CHRNA3 P32297 4/20 0.41
CHRNB1 P11230 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNB3 Q05901 1/20 0.40
HTR1D P28221 3/20 0.37
HTR1B P28222 3/20 0.37
HTR2A P28223 3/20 0.37
MEN1 O00255 3/20 0.37
MAPT P10636 3/20 0.37
KMT2A Q03164 3/20 0.37
TDP1 Q9NUW8 3/20 0.37
TP53 P04637 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
MAPK1 P28482 2/20 0.37
HSD17B10 Q99714 2/20 0.37
HPGD P15428 2/20 0.37
ALDH1A1 P00352 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7920441 0.86 MCHR1 (0.45) MCHR1HTR1DHTR1BHTR2AMEN1
Hydrochloric Acid SCHEMBL7913385 0.86 HTR1D (0.38) CHRNB4CHRNA3HTR1DHTR1BHTR2A
SCHEMBL7920434 0.82 MCHR1 (0.45) MCHR1CHRNB4CHRNA3CHRNB1CHRNB2
Oxalic Acid SCHEMBL7919986 0.78 MAPT (0.33) HTR1DHTR1BHTR2AMEN1MAPT
SCHEMBL7448439 0.77 HTR1D (0.54) HTR1DHTR1BHTR2AMEN1MAPT
SCHEMBL6927404 0.74 HTR1D (0.68) MCHR1HTR1DHTR1BHTR2AMEN1
SCHEMBL6927402 0.74 HTR1D (0.68) MCHR1HTR1DHTR1BHTR2AMEN1
SCHEMBL6928603 0.74 HTR1D (0.68) MCHR1HTR1DHTR1BHTR2AMEN1
SCHEMBL8798964 0.72 HTR1D (0.60) MCHR1HTR1DHTR1BHTR2AMEN1
SCHEMBL6927766 0.70 HTR1D (0.69) MCHR1HTR1DHTR1BHTR2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001766-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2001-04-04 EP disclosed
EP-1001766-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999001127-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-01-14 WO disclosed