SCHEMBL7920441

SCHEMBL7920441

COc1ccc(NC(=O)C2(c3noc(C)n3)C=CC(c3ccccc3C)=CC2)cc1OCCN1CCCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 7/20 0.45
HTR2A P28223 7/20 0.40
HTR2C P28335 6/20 0.40
HTR1D P28221 2/20 0.40
HTR1B P28222 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
SLC5A7 Q9GZV3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7920436 0.86 MCHR1 (0.43) MCHR1HTR2AHTR2CHTR1DHTR1B
Hydrochloric Acid SCHEMBL7913385 0.82 HTR1D (0.38) HTR2AHTR2CHTR1DHTR1BKDM4E
SCHEMBL7920439 0.80 MCHR1 (0.46) MCHR1HTR2AHTR2CHTR1DHTR1B
Oxalic Acid SCHEMBL7919986 0.79 MAPT (0.33) HTR2AHTR2CHTR1DHTR1BKDM4E
SCHEMBL7448439 0.79 HTR1D (0.54) HTR2AHTR2CHTR1DHTR1BKDM4E
SCHEMBL6921901 0.72 HTR1D (0.75) MCHR1HTR2AHTR2CHTR1DHTR1B
SCHEMBL7439830 0.72 HTR1D (0.68) MCHR1HTR2AHTR2CHTR1DHTR1B
SCHEMBL7067303 0.72 HTR1D (0.74) MCHR1HTR2AHTR2CHTR1DHTR1B
SCHEMBL29055273 0.70 HTR1D (0.39) MCHR1HTR2AHTR2CHTR1DHTR1B
SCHEMBL29055293 0.69 FGFR4 (0.42) HTR2AHTR2CHTR1DHTR1BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001766-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2001-04-04 EP disclosed
EP-1001766-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999001127-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-01-14 WO disclosed