SCHEMBL7920485

SCHEMBL7920485

COC(=O)c1ccc(C#Cc2ccc3c(c2)C(C)(C)CO3)cc1O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 5/20 0.48
RARG P13631 5/20 0.48
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
PDK2 Q15119 1/20 0.43
PDK4 Q16654 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
GAA P10253 1/20 0.41
PTPN11 Q06124 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
RARA P10276 4/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
MYC P01106 1/20 0.37
ACACB O00763 1/20 0.37
RXRA P19793 1/20 0.36
KDM4E B2RXH2 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1390724 0.83 RARG (0.44) RARBRARGRARAPTGS1PTGS2
SCHEMBL19342969 0.81 RARB (0.56) RARBRARGCA12CA1CA2
SCHEMBL29820043 0.79 CA12 (0.65) CA12CA1CA2CA7PDK2
SCHEMBL15603819 0.79 CA12 (0.65) CA12CA1CA2CA7PDK2
SCHEMBL8440033 0.79 CA12 (0.41) RARBRARGCA12CA1CA2
SCHEMBL7920809 0.79 CA12 (0.48) CA12CA1CA2CA7PDK2
SCHEMBL12432422 0.75 CA12 (0.59) CA12CA1CA2CA7PDK2
SCHEMBL8440028 0.75 RARA (0.54) RARBRARGCA12CA1CA2
SCHEMBL16744298 0.74 RARB (0.73) RARBRARGCA12CA1CA2
SCHEMBL23883732 0.74 CA12 (0.57) CA12CA1CA2CA7PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2351743-A1 BICYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-08-03 EP disclosed
WO-2010050445-A1 BICYCLIC COMPOUND 武田薬品工業株式会社 (JP) 2010-05-06 WO disclosed