SCHEMBL7920959

SCHEMBL7920959

CCCCCCCCS(=O)(=O)NCCSc1cc(F)c(OCC(=O)O)c(F)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
NFKB1 P19838 1/20 0.52
PMP22 Q01453 1/20 0.52
HIF1A Q16665 1/20 0.52
HSD17B10 Q99714 1/20 0.52
RELA Q04206 4/20 0.36
THRA P10827 3/20 0.35
THRB P10828 3/20 0.35
PLA2G4B P0C869 2/20 0.35
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34
TSHR P16473 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7920567 0.91 ALDH1A1 (0.48) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7911808 0.88 ALDH1A1 (0.41) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7911917 0.88 ALDH1A1 (0.41) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7920744 0.83 ALDH1A1 (0.48) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7918856 0.79 ALDH1A1 (0.41) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7920723 0.79 ALDH1A1 (0.41) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7919297 0.76 ALDH1A1 (0.84) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7920964 0.76 CNR2 (0.38) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7920747 0.76 CNR2 (0.38) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7920941 0.76 ALDH1A1 (0.69) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0811375-B1 GLUTAMIC ACID RECEPTOR AGONIST NIPPON SUISAN KAISHA LTD (JP) 2001-01-03 EP disclosed
US-5955505-A TREATING NERVE DEGENERATIVE DISORDERS NIPPON SUISAN KAISHA, LTD. (JP) 1999-09-21 US disclosed
EP-0811375-A1 GLUTAMIC ACID RECEPTOR AGONIST NIPPON SUISAN KAISHA, LTD. (JP) 1997-12-10 EP disclosed
EP-0469901-B1 Sulfonamide derivatives TAISHO PHARMACEUTICAL CO LTD (JP) 1994-10-19 EP disclosed
US-5189211-A Thromboxane A2 antagonists TAISHO PHARMACEUTICAL CO., LTD. (JP) 1993-02-23 US disclosed
EP-0469901-A1 Sulfonamide derivatives TAISHO PHARMACEUTICAL CO. LTD (JP) 1992-02-05 EP disclosed