SCHEMBL7920993

SCHEMBL7920993

NC(=O)COc1c(F)cc(SCCN(O)S(=O)(=O)c2ccc(Cl)cc2)cc1F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
NFKB1 P19838 1/20 0.53
PMP22 Q01453 1/20 0.53
HIF1A Q16665 1/20 0.53
HSD17B10 Q99714 1/20 0.53
HTT P42858 2/20 0.39
PKM P14618 1/20 0.39
KMT2A Q03164 3/20 0.35
ACLY P53396 1/20 0.35
NPC1 O15118 1/20 0.34
CXCR3 P49682 1/20 0.34
MAPT P10636 4/20 0.33
CA12 O43570 3/20 0.33
CA1 P00915 3/20 0.33
CA2 P00918 3/20 0.33
CA4 P22748 3/20 0.33
CA9 Q16790 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7919292 0.90 ALDH1A1 (0.66) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7924029 0.89 ALDH1A1 (0.41) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7920584 0.80 ALDH1A1 (0.81) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7911824 0.79 ALDH1A1 (0.52) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL18377181 0.78 ALDH1A1 (0.65) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL20383348 0.78 ALDH1A1 (0.65) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7918887 0.78 ALDH1A1 (0.52) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL20387769 0.76 ALDH1A1 (0.62) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL18377183 0.74 ALDH1A1 (0.60) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7919298 0.73 DAGLA (0.41) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0811375-B1 GLUTAMIC ACID RECEPTOR AGONIST NIPPON SUISAN KAISHA LTD (JP) 2001-01-03 EP disclosed
US-5955505-A TREATING NERVE DEGENERATIVE DISORDERS NIPPON SUISAN KAISHA, LTD. (JP) 1999-09-21 US disclosed
EP-0811375-A1 GLUTAMIC ACID RECEPTOR AGONIST NIPPON SUISAN KAISHA, LTD. (JP) 1997-12-10 EP disclosed
EP-0469901-B1 Sulfonamide derivatives TAISHO PHARMACEUTICAL CO LTD (JP) 1994-10-19 EP disclosed
US-5189211-A Thromboxane A2 antagonists TAISHO PHARMACEUTICAL CO., LTD. (JP) 1993-02-23 US disclosed
EP-0469901-A1 Sulfonamide derivatives TAISHO PHARMACEUTICAL CO. LTD (JP) 1992-02-05 EP disclosed