SCHEMBL7920997

SCHEMBL7920997

O=C(COc1c(F)cc(SCCNS(=O)(=O)c2ccc(Cl)cc2)cc1F)NO

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.64
CYP1A2 P05177 1/20 0.64
CYP3A4 P08684 1/20 0.64
CYP2C9 P11712 1/20 0.64
NFKB1 P19838 1/20 0.64
PMP22 Q01453 1/20 0.64
HIF1A Q16665 1/20 0.64
HSD17B10 Q99714 1/20 0.64
MAPT P10636 2/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
LMNA P02545 2/20 0.47
HTT P42858 2/20 0.47
MMP1 P03956 1/20 0.45
MEP1B Q16820 1/20 0.45
TSHR P16473 2/20 0.44
GAA P10253 1/20 0.44
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2925987 0.90 ALDH1A1 (0.69) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7919293 0.90 ALDH1A1 (0.79) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7924034 0.89 ALDH1A1 (0.57) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7920584 0.89 ALDH1A1 (0.81) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7918789 0.88 ALDH1A1 (0.64) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7911825 0.86 ALDH1A1 (0.62) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7911552 0.85 ALDH1A1 (0.61) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7924024 0.85 ALDH1A1 (0.60) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL5142189 0.82 ALDH1A1 (0.59) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1
SCHEMBL7919257 0.81 ALDH1A1 (0.69) ALDH1A1CYP1A2CYP3A4CYP2C9NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0811375-B1 GLUTAMIC ACID RECEPTOR AGONIST NIPPON SUISAN KAISHA LTD (JP) 2001-01-03 EP disclosed
US-5955505-A TREATING NERVE DEGENERATIVE DISORDERS NIPPON SUISAN KAISHA, LTD. (JP) 1999-09-21 US disclosed
EP-0811375-A1 GLUTAMIC ACID RECEPTOR AGONIST NIPPON SUISAN KAISHA, LTD. (JP) 1997-12-10 EP disclosed
EP-0469901-B1 Sulfonamide derivatives TAISHO PHARMACEUTICAL CO LTD (JP) 1994-10-19 EP disclosed
US-5189211-A Thromboxane A2 antagonists TAISHO PHARMACEUTICAL CO., LTD. (JP) 1993-02-23 US disclosed
EP-0469901-A1 Sulfonamide derivatives TAISHO PHARMACEUTICAL CO. LTD (JP) 1992-02-05 EP disclosed