SCHEMBL7921240

SCHEMBL7921240

Cc1csc(-c2cccs2)c1Br

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
RAB9A P51151 6/20 0.36
KDM4E B2RXH2 6/20 0.36
NPC1 O15118 5/20 0.36
ALDH1A1 P00352 5/20 0.36
SMN1; SMN2 Q16637 4/20 0.36
TDP1 Q9NUW8 4/20 0.35
MAPT P10636 4/20 0.35
HPGD P15428 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CASP3 P42574 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4614749 0.82 MEN1 (0.39) MEN1KMT2ARAB9AKDM4ENPC1
SCHEMBL7760837 0.80 MEN1 (0.38) MEN1KMT2ARAB9AKDM4ENPC1
SCHEMBL4586849 0.78 MEN1 (0.37) MEN1KMT2ARAB9AKDM4ENPC1
SCHEMBL10086063 0.76
SCHEMBL4613684 0.73 MAPT (0.34) MEN1KMT2ARAB9AKDM4ENPC1
Anthracene SCHEMBL28886884 0.73 RPS6KB2 (0.46) MEN1KMT2ARAB9AKDM4ENPC1
SCHEMBL3061563 0.73 MEN1 (0.33) MEN1KMT2ARAB9AKDM4ENPC1
SCHEMBL992407 0.72 ALDH1A1 (0.36) MEN1KMT2ARAB9AKDM4ENPC1
SCHEMBL4149778 0.72 MAPT (0.33) MEN1KMT2ARAB9AKDM4ENPC1
SCHEMBL723960 0.71 CYP2A6 (0.44) MEN1KMT2ARAB9AKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6274590-B1 ADMINISTERING 3,4-DIARYLTHIOPHENE DERIVATIVE TO TREAT ECZEMA, BURNS, PSORIASIS, AND DERMATITIS G. D. SEARLE & CO. 2001-08-14 US disclosed