SCHEMBL7922009

SCHEMBL7922009

NC(=O)C1=Cc2ccccc2S(=O)(=O)CC1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
L3MBTL1 Q9Y468 3/20 0.32
MAPK1 P28482 1/20 0.32
LMNA P02545 1/20 0.31
HSD17B10 Q99714 2/20 0.31
POLB P06746 1/20 0.31
CYP3A4 P08684 1/20 0.31
PARP1 P09874 1/20 0.31
MAPT P10636 1/20 0.31
TSHR P16473 1/20 0.31
CYP2C19 P33261 1/20 0.31
RECQL P46063 1/20 0.31
BLM P54132 1/20 0.31
PMP22 Q01453 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7931055 0.98 MEN1 (0.37) MEN1KMT2AL3MBTL1MAPK1LMNA
Hydrochloric Acid SCHEMBL7922067 0.84 MAPK1 (0.34) MEN1KMT2AL3MBTL1MAPK1LMNA
SCHEMBL7922036 0.83 MEN1 (0.37) MEN1KMT2AL3MBTL1MAPK1LMNA
SCHEMBL7378111 0.78
SCHEMBL7922065 0.71 NOTUM (0.41) TSHR
SCHEMBL950483 0.70 KDM1A (0.43) L3MBTL1HSD17B10POLBCYP3A4PARP1
SCHEMBL8651466 0.69 ALOX5 (0.38) L3MBTL1LMNAHSD17B10POLBCYP3A4
SCHEMBL7526631 0.67 MEN1 (0.43) MEN1KMT2AL3MBTL1MAPK1LMNA
SCHEMBL5655529 0.67 MEN1 (0.33) MEN1KMT2AL3MBTL1MAPK1LMNA
SCHEMBL30219251 0.67 PARP1 (0.44) MAPK1LMNAHSD17B10PARP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP claimed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO claimed
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed