SCHEMBL7922186

SCHEMBL7922186

COc1ccc(NC(=O)c2ccc(-c3ccccc3)cc2Cl)cc1OCCN(C)C

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 11/20 0.69
KDR P35968 5/20 0.60
HTR2C P28335 2/20 0.55
HDAC8 Q9BY41 1/20 0.53
NR1H4 Q96RI1 1/20 0.49
HTR1D P28221 2/20 0.49
HTR1B P28222 2/20 0.49
HTR2A P28223 2/20 0.49
KDM4E B2RXH2 1/20 0.49
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
MAPT P10636 1/20 0.49
HPGD P15428 1/20 0.49
ALOX15 P16050 1/20 0.49
MAPK1 P28482 1/20 0.49
KMT2A Q03164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7678814 0.91 MCHR1 (0.73) MCHR1KDRHTR2CNR1H4HTR1D
SCHEMBL6928640 0.86 MCHR1 (0.92) MCHR1HTR2CHTR1DHTR1BHTR2A
SCHEMBL6927547 0.83 MCHR1 (0.75) MCHR1KDRHTR2CHTR1DHTR1B
SCHEMBL7646291 0.82 MCHR1 (0.74) MCHR1KDRHTR2C
SCHEMBL6920493 0.81 MCHR1 (0.76) MCHR1KDRHTR2CHTR1DHTR1B
SCHEMBL6926020 0.81 MCHR1 (0.80) MCHR1HTR2C
SCHEMBL6927530 0.80 MCHR1 (0.76) MCHR1KDRHTR2CHTR1DHTR1B
SCHEMBL6927561 0.80 MCHR1 (0.76) MCHR1KDRHTR2CHTR1DHTR1B
SCHEMBL7670306 0.79 MCHR1 (0.77) MCHR1HTR2C
SCHEMBL6927709 0.78 MCHR1 (0.77) MCHR1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001766-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2001-04-04 EP disclosed
EP-1001766-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999001127-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-01-14 WO disclosed