SCHEMBL7922358

SCHEMBL7922358

CC(C)(C)OC(=O)NC1=NC2(c3cc([N+](=O)[O-])ccc3F)COC[C@@H](F)[C@H]2CS1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.35
BACE1 P56817 12/20 0.35
BACE2 Q9Y5Z0 11/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
THRB P10828 1/20 0.35
HTT P42858 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.34
GNRHR P30968 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9913123 1.00 DRD2 (0.35) DRD2BACE1BACE2ALDH1A1GAA
SCHEMBL9913133 0.94 DRD2 (0.35) DRD2BACE1BACE2ALDH1A1GAA
SCHEMBL9913132 0.94 DRD2 (0.35) DRD2BACE1BACE2ALDH1A1GAA
SCHEMBL7925298 0.94 DRD2 (0.35) DRD2BACE1BACE2ALDH1A1GAA
SCHEMBL9913143 0.92 BACE1 (0.35) DRD2BACE1BACE2ALDH1A1GAA
SCHEMBL7916603 0.92 BACE1 (0.35) DRD2BACE1BACE2ALDH1A1GAA
SCHEMBL8030093 0.90 BACE1 (0.44) DRD2BACE1BACE2ALDH1A1GAA
SCHEMBL13009269 0.90 BACE1 (0.44) DRD2BACE1BACE2ALDH1A1GAA
SCHEMBL2632338 0.88 BACE1 (0.45) DRD2BACE1BACE2ALDH1A1GAA
SCHEMBL10288946 0.88 BACE1 (0.45) DRD2BACE1BACE2ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038686-A1 NOVEL FUSED AMINODIHYDROTHIAZINE DERIVATIVE エーザイ・アール・アンド・ディー・マネジメント株式会社 (JP) 2010-04-08 WO disclosed