SCHEMBL7922547

SCHEMBL7922547

Bc1cc(F)c(C(=O)Nc2cnc(C3=C(C)CCN(c4ncccc4F)C3)cn2)c(F)c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.40
IL2 P60568 11/20 0.39
TRPV1 Q8NER1 4/20 0.38
STIM1 Q13586 1/20 0.37
ORAI1 Q96D31 1/20 0.37
ORAI2 Q96SN7 1/20 0.37
GRM4 Q14833 1/20 0.34
HTR1A P08908 1/20 0.33
HTR1B P28222 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR1F P30939 1/20 0.33
HTR2B P41595 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3374258 0.93 IL2 (0.40) HDAC6IL2TRPV1STIM1ORAI1
Hydrochloric Acid SCHEMBL1782166 0.92 IL2 (0.39) HDAC6IL2TRPV1STIM1ORAI1
SCHEMBL7922608 0.92 IL2 (0.43) HDAC6IL2TRPV1STIM1ORAI1
SCHEMBL1781058 0.92 HDAC6 (0.40) HDAC6IL2TRPV1STIM1ORAI1
Hydrochloric Acid SCHEMBL614560 0.91 IL2 (0.43) HDAC6IL2TRPV1STIM1ORAI1
SCHEMBL1780826 0.90 IL2 (0.38) HDAC6IL2TRPV1STIM1ORAI1
SCHEMBL1782159 0.87 IL2 (0.42) HDAC6IL2TRPV1STIM1ORAI1
SCHEMBL7920820 0.85 STIM1 (0.44) IL2TRPV1STIM1ORAI1ORAI2
SCHEMBL614875 0.85 IL2 (0.43) HDAC6IL2TRPV1STIM1ORAI1
SCHEMBL7914099 0.85 IL2 (0.41) IL2TRPV1STIM1ORAI1ORAI2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010039236-A1 COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2010-04-08 WO disclosed